РектАктив®

General characteristics. Structure:

Active agent: A horse-chestnut of fruits of extract of the dry, containing 20% of the sum of triterpenovy saponins in terms of эсцин 50 mg or 100 mg. Excipient: Fatty acids of glycerides (Vitepsola of N 15, Fat firm) enough for receiving suppository weighing 1,0 g.

Description: 

Suppositories dosage of 50 mg of light brown color of a torpedo-shaped form. Suppositories dosage of 100 mg of brown color of a torpedo-shaped form. On a surface and on a cut of suppositories impregnations of dark brown color are allowed.

Pharmacological properties:

Triterpenovy saponin эсцин, contained in extract of a horse-chestnut stimulates interoretseptor of a mucous membrane of a rectum, causing strengthening of its vermicular movement and bystry evacuation of fecal masses. The effect occurs in 5-15 min. after suppository use. Desires to bowel emptying stop after the act of defecation. Drug does not cause stretching of walls of a rectum, strengthens and tones up smooth muscles of this body. At course use drug recovers a defecation reflex and normalizes a defecation biorhythm.

Indications to use:

Locks: functional (usual, senile, locks at slow-moving patients, the locks connected with decrease in sensitivity of the receptor device of a rectum and disturbance of a biorhythm of defecation).

Route of administration and doses:

Drug is used rektalno (enter into a rectum) 1 time a day in 5-15 min. prior to the planned act of defecation. To take out suppository from a strip packaging, to break off one cell with suppository on a notch and having separated edges of a tape to pull for them in different directions. To enter suppository into an anus the pointed end, whenever possible deeply. For more convenient administration of suppository it is recommended to bend down, sit down on hunkers or to lay down sideways, having drawn in legs.

Single dose for adult 50-100 mg of 1 times a day; the maximum single dose – 300 mg; the maximum daily dose – 300 mg. Duration of treatment is no more than 30 days. Further treatment by drug perhaps only after consultation with the doctor.

Side effects:

Allergic reactions, short-term burning sensation in a rectum are in some cases possible.

Contraindications:

Hypersensitivity, intestinal impassability, acute inflammatory diseases of abdominal organs, acute hemorrhoids, acute proctitis and paraproctitis, spastic lock, tumors and cracks of a rectum.

Pregnancy and breastfeeding: 

Use of drug during the periods of pregnancy and a lactation is possible only when the potential advantage for mother exceeds risk for a fruit and the baby.

Storage conditions:

In the dry place protected from light at a temperature not above 25 °C. To store in the place, unavailable to children.

Period of validity: 1 year 10 months. Not to use after a period of validity.

Issue conditions:

According to the recipe

Packaging:

Suppositories rectal 50 mg and 100 mg. On 1 and on 5 suppositories in a blister strip packaging from a film polyvinyl chloride. On 1 planimetric packaging with 1 suppository in a cardboard insert. On 2 cardboard inserts together with the application instruction in a pack cardboard. On 1 or on the 2nd blister strip packagings with 5 suppositories together with the application instruction in a pack cardboard.