Baralgetas

Baralgetas – the non-narcotic combined means killing pain and spasms.

Form of release and structure

Dosage forms of drug:

• Tablets (on 10 pieces in blisters, 1 or 10 blisters in a pack cardboard);
• Solution for intramuscular and intravenous administration (in ampoules of dark glass, in a pack of cardboard 5 ampoules).

Content of active agents is to 1 tablet/ampoule of Baralgetas:

• Metamizole sodium – 500 mg;
• Pitofenona a hydrochloride – 5 mg;
• Fenpiveriniya bromide – 0,1 mg.

Metamizole sodium has febrifugal and soothing effect, a fenpiveriniya bromide and a pitofenona a hydrochloride relax smooth muscles of internals. Action of a pitofenon of a hydrochloride is similar to action of a papaverine.

Indications to use

Baralgetas's use is recommended at the moderate and mild pains caused by spasms of muscles of internals (spasms of a bladder and ureters, renal, intestinal and bilious gripes).

Baralgetas's appointment is effective also at dyskinesia of bile-excreting channels, chronic colitis, algodismenory, a postcholecystectomy syndrome, diseases of bodies of a small pelvis.

Anesthetic can be used in short therapy of a mialgiya, ischialgia, arthralgia, neuralgia and as soothing after operations and diagnostic procedures.

Contraindications

• Oppression of the hemopoietic function of marrow;
• Serious renal and liver failure;
• Tachyarrhythmia, stenocardia, dekompensirovanny heart chronic failure;
• Closed-angle glaucoma;
• Prostate hyperplasia;
• Impassability of intestines;
• Collapse;
• Hypersensitivity;
• Pregnancy, lactation.

Intravenously do not administer the drug to children up to 3 months or weighing less than 5 kg.

Tablets are contraindicated to children up to 5 years.

With caution Baralgetas it is necessary to take at a liver and renal failure, bronchial asthma, tendency to the lowered pressure, hypersensitivity to anti-inflammatory nonsteroid drugs.

Route of administration and dosage

Tablets

The recommended dosing for various age groups:

• Children of 5-7 years: a single dose – ^1/2 tablets, maximum daily – 2 tablets;
• Children of 8-11 years: one-time – ^1/2 tablets, maximum daily – 4 tablets;
• Children of 12-14 years: one-time – 1 tablet, maximum daily – 6 tablets;
• Teenagers are more senior than 15 years and adults: a single dose –1-2 tablets, frequency rate of reception – 2-3 times a day.

Solution for intramuscular and intravenous administration

Intravenously the drug is administered to teenagers 15 years and the adult are more senior at heavy and acute gripes – in number of 2 ml. It is necessary to enter Baralgetas slowly, on 1 ml for 1 minute. If necessary solution can be entered once again – in 6-8 h. Intramusculary Baralgetas enter 2-3 times a day 2-5 ml. An admissible daily dose – 10 ml, treatment duration – 5 days.

Children can administer the drug as anesthetic intramusculary and intravenously according to age:

• 3-11 months: of 0,1-0,2 ml and only intramusculary;
• 1-2 years: 0,2-0,3 ml intramusculary or 0,1-0,2 ml intravenously;
• 3-4 years: 0,3-0,4 ml intramusculary or 0,2-0,3 ml intravenously;
• 5-7 years: 0,4-0,5 ml intramusculary or 0,3-0,4 ml intravenously;
• 8-12 years: 0,6-0,7 ml intramusculary or 0,5-0,6 ml intravenously;
• 12-15 years: 0,8-1,0 ml intramusculary or intravenously.

Before an injection the ampoule with drug should be taken in a hand to warm solution to room temperature.

Side effects

• Allergic reactions: small tortoiseshell, Quincke's disease, erythema, epidermal toxic necrolysis, bronchospasm, acute anaphylaxis;
• Urinary system: disturbance of renal function, anury, proteinuria, oliguria, nephrite, urine discoloration;
• Bodies of a hemopoiesis: agranulocytosis, leukopenia, thrombocytopenia;
• Cardiovascular system: lowering of arterial pressure;
• Anticholinergic effects: tachycardia, accommodation paresis, dryness mucous a mouth, the complicated urination, reduced sweating;
• Local reactions: at introduction in oil infiltrates in an injection site are possible.

At overdose vomiting, drowsiness, nausea, pain in epigastriums, pressure decrease, disturbance of renal and hepatic function, a spasm develops. In these cases to the patient wash out a stomach, allow to drink absorbent carbon.

Special instructions

During Baralgetas's use it is not necessary to use the substances containing ethanol.

In case of long (more than one week) reception of a medicine it is necessary to control a functional condition of a liver and a picture of peripheral blood.

It is impossible to accept Baralgetas for stopping of an acute pain in a stomach before identification of its reason.

It is necessary to stop immediately drug intake at suspicion on an agranulocytosis, and also in case of detection of thrombocytopenia.

The feeding women have to interrupt breastfeeding for the period of treatment.

Baralgetas's use by children up to 5 years and the patients receiving cytostatic drugs has to be carried out under observation of the doctor.

For intramuscular introduction it is necessary to use a long fine needle.

Has no clinical value probable coloring of urine in red color (allocation of a metabolite).

Occupations potentially dangerous types of works, control of difficult mechanisms, motor transport it is necessary to make with care as the speed of mental and physical reaction can be reduced.

Analogs

The drugs similar to Baralgetas on the active operating components: Took, Bralangin, Maksigan, Plenalgin, Revalgin, Renalgan, Spazgan, Spazmalgon, Spazmalin, Spazmoblok, Spazmogard, Trinalgin, the Geomagician.

The analogs close on the influence mechanism: Akofil, Analgin, Andipal, Antipirin, Baralgin of M, Benalgin, Kvintalgin, Pentabufen, Pentalgin, Santoperalgin, Sedal-M, Sedalgin-Neo, Tempalgin, Tempanginol, Tetralgin, Kvatroks.

Terms and storage conditions

To store in the dry place protected from light, at the room temperature not above 25 °C.

Period of validity – 5 years.